Cabergoline dostinex in bodybuilding how to accept reviews

Author: Yuri Klimishin - an iron lover and a veteran of the “chemical” front. Place in the ranking of authors: 2

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2014-12-09
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Important! The “Your Trainer” website does not sell or encourage the use of anabolic steroids and other potent substances. The information is provided so that those who decide to take them do so as competently as possible and with minimal risk to health.

Medicines from both groups are very useful to the user of anabolic steroids. This refers to people who take a thoughtful approach to building the healthy body of their dreams. But you need to use these helpers correctly and on time, otherwise they will easily turn from friends into enemies.

Very often, amateurs really underestimate all the pitfalls of these drugs. Meanwhile, the side effects of both the first and second are much more dangerous and global than the side effects of the same anabolic steroids. But you won’t be able to do without them completely either. So there is only one way out - to use them correctly.

Harm from excessive levels of prolactin in the body

Initially, you should understand what prolactin is . This is a hormone that has a direct effect on the ability to reproduce. Elevated levels of prolactin in men negatively affect their sex life and can even cause infertility.

These negative consequences can, over time, develop into psychological problems, which can provoke apathy.

In women, the effect of the hormone is almost the same, since it affects fertility or lactation. However, we should not forget that prolactin is a female hormone and it is necessary for the normal functioning of a large number of processes occurring in the body, especially those related to childbirth and related things (bearing a fetus, breastfeeding a child).

Males do not need this hormone at all, and its increased content can be a serious problem for a bodybuilder, since lethargy and bad mood are often present, and during training or competitions there is no will to win. And as you know, the internal state is very important for success in bodybuilding, as well as in most other areas of human life.

Effect on the body

Cabergoline is known for its ability to reduce prolactin levels, which results in the removal of excess fluid and muscle gain. Bodybuilders use the drug to block side effects from the use and use of steroids. At its core, Cabergoline resembles the structure of growth hormone.

The purpose of the drug is to influence the physical condition by improving the hormonal levels of athletes. As mentioned above, Cabergoline helps to gain lean muscle mass, which is so necessary for bodybuilders.

But it is important to note that the drug is also often used for: suppression of lactation after childbirth, idiomatic hyperprolactinemia, amenorrhea, and also as one of the methods of treating Parkinson's disease.

Reasons for increasing the amount of prolactin in the body

Before considering the benefits of taking cabergoline, you should understand the reasons for the increase in prolactin.

They can be divided into two categories: related or not related to taking drugs for athletes.

Let's start with the reasons not related to taking steroids:

• diseases of the pituitary gland and hypothalamus;
• thyroid problems;
• kidney disease;
• liver diseases;
• lupus erythematosus, arthritis and other autoimmune diseases;
• low content of vitamin B6 in the body;
• a large amount of progesterone, estradiol;
• frequent stress.

It should be noted that due to the presence of congenital diseases, an increase in prolactin is not observed .

Among bodybuilders, the cause of such problems, in most cases, is illiterate use of steroids.

Particular attention should be paid to the following drugs when taking:

• Nandrolone;
• Trenbolone;
• Oxymetholone;
• Boldenone;
• other progestins.

It makes no sense to go into details about the increase in prolactin due to taking progestins, you just need to take into account some facts:

1. It is imperative to undergo hormonal tests before taking such medications. If an increased level of prolactin is observed before using the drug, then you should not resort to taking progastins.
2. While taking medications, it is necessary to carefully monitor the hormone levels, even if the dosage is small.
3. A few weeks after the start of the course, depending on the half-life (the speed at which the drug starts working), you should be tested for prolactin levels. If it is elevated, you should start taking cabergoline immediately as it eliminates the side effects of these steroids.

Sometimes, in men, prolactin increases due to excess adipose tissue. In these cases, fat deposits appear in places characteristic of the female body. Research shows that cabergoline can help such people; they just need to start bodybuilding and, after the first successes appear, start using cabergoline.

Prolactin inhibitors

Cabergoline (Dostinex) is a new generation prolactin inhibitor. It selectively stimulates dopamine type D-2 receptors. That is, it will quickly and confidently reduce the amount of excess prolactin. The most important thing is that as long as cabergoline works, previously suppressed dopamine will be restored. A reasonable dose of cabergoline is 250 mcg every four days (roughly speaking, one tablet containing 500 mcg per week). Now analogues of Dostinex have appeared and it is quite possible to use them.

Side effects of this substance (if the specified dose is observed) manifest themselves in the form of insomnia and suppressed appetite. Less commonly, deterioration in mood may occur. Not everyone has them and usually go away within a few days after starting use.

Bromocriptine (Parlodel) is also a prolactin inhibitor and is also very effective. The action is similar to cabergoline, only unlike the latter, bromine is able to somewhat inhibit the production of growth hormone by the pituitary gland (this fact has not been fully proven, but it is still worth taking into account). Another difference is the pronounced side effects. Common symptoms associated with this substance are: nausea, complete loss of appetite and migraines. Sometimes bromocriptine causes attacks of low blood pressure (which worsens all of the above side effects and causes drowsiness and physical weakness).

The most loyal way to take this medicine is to take half a tablet daily before bed and within ten days, increase to two tablets daily. One before breakfast and one before bed. This refers to tablets containing 2.5 mg of active substance.

And now the most important thing. Prolactin is a very necessary hormone in the male body. In addition to water-salt metabolism, it takes part in the formation of sperm and ensuring orgasm. But most importantly, it has an immunomodulatory effect. If we only slightly lower the natural level of prolactin, we risk permanently undermining the protective functions of our beloved body. Moreover, not only general immunity suffers, but also cellular immunity.

Benefits of consuming cabergoline

Cabergoline reduces the amount of prolactin , so people involved in bodybuilding are highly recommended to take this substance. In addition, cabergoline increases the amount of testosterone present in the male body, which significantly affects the quality of training.

Taking this substance guarantees the following effects:

• the man is unable to make concessions to his rivals, self-confidence noticeably grows;
• the woman becomes more confident and decisive, and is able to devote more effort to training.

Among other things, the use of cabergoline provides pleasant additions: reducing the time between sexual intercourse, improving sex life and, in relation to men, enlarging the penis and testicles.

Why is cabergoline needed in bodybuilding?

Athletes who take anabolic steroids often experience symptoms of gynecomastia. This is a serious disease caused by hormonal imbalance; it is expressed not only in the growth of the mammary glands, but is also manifested by the presence of lactation. In a man, when the nipple is squeezed, a small amount of fluid may be released. This symptom indicates hormonal imbalances. Usually this is an imbalance between estrogens, prolactin and medications. When symptoms appear, you need to adjust the dosage of anabolic steroids, and also use cabergoline if the concentration of prolactin increases.

Features of the use of cabergoline

If cabergoline is taken in parallel with the use of progestins, then the dosage is as follows - 0.25 milligrams once every 4 days (with elevated prolactin levels, once every 2 days). In addition, in such a situation, the product helps relieve swelling from the muscles and face, fluid retention in the tissues is significantly reduced, which increases the growth of lean muscles.

Cabergoline can be used without drugs with progestin activity, which improves the quality of life and results after completing the course. In this case, the dosage is as follows: 0.5 milligrams once every ten days.

Some athletes wish to increase their performance without resorting to AAC. The drug can help them too. However, it should be noted that for these purposes it is necessary to significantly reduce the dosage .

A common mistake is to lower prolactin too much. This leads to sleep disturbances, poor mood, poor appetite, or even decreased immunity. To recover from this, you need to stop taking the drug for some, sometimes long, time (wait until it stops working) and then reduce the frequency of use and reduce the dosage.

Dostinex in bodybuilding can be used on PCT if prolactin is too high.

Cabergoline is a hormonal agent. Therefore, while taking this drug, you must take the same precautions as with most similar medications:

• dosage must be observed;
• take exactly by the hour;
• seek help from specialists at the slightest side effects;
• strictly follow the instructions and do not skip taking the product.

Pharmacological properties of cabergoline for men

The drug acts as an agonist of dopamine type receptors. The active substance is a derivative of ergoline, which allows it to have a strong prolactin-lowering effect. Cabergoline acts on dopamine receptors, which reduces the concentration of prolactin in the blood. The effectiveness of the drug is noticeable just three hours after use.

When cabergoline is used by men, it does not affect other hormones. The only associated effect is a decrease in blood pressure.

Cabergoline: analogues

Many bodybuilders may be confused by the large number of names for cabergoline. Don't be afraid , the differences are only external .

Whatever the name of cabergoline analogues, they are all characterized by high quality of action.

There are the following varieties of cabergoline , which can be purchased at the pharmacy:

1. Bergolak - manufacturer Russia. Contains 8 tablets of 0.5 milligrams.
2. Cabaser is manufactured in Italy by Pfizer. Tablet - 1 milligram of active ingredient.
3. Agaltex - manufacturer Czech Republic. Contains the active substance, in the amount of 2 or 8 pieces of 0.5 milligrams.
4. Alacting - the form and composition are identical to Agaltex. Manufacturer: Teva.
5. Dostinex - manufacturer Italy, Pfizer company. Contains 8 tablets of 0.5 mg each. The composition of the drug Dostinex is as follows: cabergoline, lactose, leucine.
6. Kaberlin. Contains 2 tablets of 0.25 mg or 8 tablets of 0.25 mg. Caberline is the least popular analogue of cabergoline.

Drugs with other names may appear, since they are very relevant and many manufacturers buy licenses for the production of cabergoline.

Difference between cabergoline and Dostinex

Some people ask the question: “Which is better Cabergoline or Dostinex?” . It is very easy to answer - Dostinex is cybergolin. Dostinex is simply the best of all analogues.

What brands is it sold under?

Despite the fact that the rights to the Cabergoline trademark belong to the American company Pharmacia, today this drug is produced in many countries, and a huge number of its names are known. Here are the most common of them:

• Dostinex is the second most popular name for Cabergoline, manufactured by the Italian company Pfizer;
• Bergolak - produced in Russia;
• Cabacer - made in Italy;
• Agalates - made in the Czech Republic;
• Alakting is a form of Agaltex, which is also manufactured in Czech factories.

Overdose symptoms

Studies show that the use of high dosages of cabergoline (more than 0.5 mg per day) leads to the development of a large number of side effects:

• digestive system disorders (the most common option): constipation, dyspepsia, nausea;
• problems with the cardiovascular system;
• nervous diseases: depression, distortion of consciousness, insomnia;
• negative reaction of the immune system (rare): hypersensitivity, skin rash;
• disorder of the hematopoietic system (rare);
• problems with the respiratory system: nosebleeds, shortness of breath, pulmonary fibrosis.

It has been noticed that if you do not exceed the dosage , then negative effects are very rare or absent at all.

On forums related to this topic, the most common messages are about poor appetite and loss of mood. A simple conclusion follows from this - you must adhere to absolutely all instructions and monitor your condition very carefully. Then there will be no problems. However, before you start using cabergoline, you should consult your doctor about this.

What side effects are possible when using Cabergoline?

In sports, the drug is considered safe, although it has some side effects.
The most common symptoms reported in the studies were headache (26 percent), nausea (27 percent), and vomiting. The latter negative effect was recorded in only two percent of subjects. It should also be noted that other side effects are possible, but they are extremely unlikely. All negative properties of Dostinex are directly related to the dosages used. This suggests that you should start taking the drug with a minimum dose and increase it if necessary.

Contraindications

It should not be used by pregnant women, lactation, psychosis, respiratory dysfunction, fibrosis, liver problems, hypertension, heart disorders, preeclampsia, or hypersensitivity to the components of the drug.

Professionals recommend taking the medication prescribed by the doctor. Before use, contraindications should be excluded to avoid side effects. Athletes using the medicine in reduced quantities rarely experience complications. More often, bodybuilders talk about the problem of depressed mood and loss of appetite.

They are necessary to eliminate the side effects of estrogen and progestogen types.

However, they must be used in strict accordance with the instructions, since they are not without their own negative properties.

Aromatization - what is it?

This process is the conversion of male hormones into estrogens. Aromatization occurs in the body of every man and is necessary to maintain the required hormonal balance. However, during the use of some AAS, this biochemical reaction will sharply accelerate. Aromatizing anabolics include all Testosterone-based drugs, as well as Methandienone, Methyltestosterone, Oxymetholone and Boldenone.

If you do not order aromatase inhibitors when using them. then you will probably encounter gynecomastia and active fluid retention in the body. It should be noted that among all the AAS noted above, Boldenone aromatizes less than other drugs. As a result, in his solo course, aromatase inhibitors are used only by those athletes whose bodies have a tendency to develop estrogenic side effects.

Reasons for aromatization

Now we will consider only those cases that can be provoked by the use of AAS:

• The use of aromatizing anabolic steroids in high doses. To avoid health problems, athletes need to start using the drug in small quantities. You can increase doses and switch to combined courses only after the body adapts to the work of light steroids and the effectiveness of their use decreases.
• Problems with liver function. If you carry out the course correctly, but symptoms of estrogen-type side effects still appear, then you need to urgently check your liver.
• High concentration of aromatase enzyme in the body. In such a situation, it is not worth using AAS that are prone to aromatization at all.

There are two classes of antiestrogens used in sports:

• Aromatase inhibitors.
• Estrogen receptor blockers.

Now we will talk about all these medications and the rules for their use.

Aromatase inhibitors

Proviron

It is a strong androgen with antiestrogenic properties. Compared to other aromatase inhibitors, it is less effective. However, in light courses, Mesterolone (the active ingredient of Proviron) copes with its task perfectly. It is also worth saying that the price of this anti-estrogen is low, which has a positive effect on its popularity.

The recommended daily dosage of Proviron is 25-50 mg. Anti-estrogen is used in higher quantities by professional bodybuilders during the cutting period. In addition to the ability to inhibit the aromatase enzyme, Mesterolone allows you to give extra hardness to the muscles, because it is a strong androgen. This is why you should not exceed the recommended dosage.

Anastrozole

The most famous third generation aromatase inhibitor. This drug is able to suppress the aromatization process in a short time, which will lead to a decrease in the concentration of female hormones. Note that all aromatase inhibitors are used directly on an anabolic cycle before the start of PCT.

It is necessary to take Anastrozole every second day, 0.5 mg. Some athletes begin to use it only when first symptoms of estrogenic negative effects appear. In this case, take 1 mg immediately, and then 0.5 mg every other day until the side effects completely disappear. Since this is a medication, an overdose can cause negative effects. Among them it is worth noting:

• Depression.
• A sharp drop in appetite.
• Sleep disturbances.
• decreased sexual desire.
• Bone pain.

All of them are associated with a drop in estrogen concentrations below the minimum permissible limits. For the normal functioning of the male body, it must contain estrogen in a certain amount.

Exemestane and Letrozole

These drugs are similar to Anastrozole in terms of effectiveness. However, the drug discussed above is much more popular among athletes, since when taking it, potential side effects can be controlled.

Cytadren (Aminoglutethimide)

This drug is not only a powerful anti-estrogen, but also has strong anti-catabolic properties. However, after the appearance of Anastrozole on the market, Cytadren practically ceased to be used by athletes, as it has a large list of side effects.

Testolactone

This is the most advanced aromatase inhibitor, superior to all medications discussed above not only in terms of effectiveness but also safety. However, its price is extremely high.

When using aromatase inhibitors, you need to follow two rules:

• Use them only on an anabolic cycle before starting PCT.
• If aromatase inhibitors in recommended dosages do not allow you to avoid estrogenic side effects, then you need to check your liver or reduce the dose of AAS.

Estrogen receptor blockers

Three medications belong to this class of antiestrogens:

• Toremifene.
• Clomid.
• Tamoxifen.

They are used only during the period of rehabilitation therapy after anabolic courses. The only exception here is Tamoxifen, which can help get rid of lumps in the nipple area. Aromatase inhibitors cannot solve this problem. These drugs may also help when using Oxymetholone. This anabolic does not aromatize, but helps increase the activity of estrogen receptors.

Consequences of high prolactin levels

Trenbolones, Nandrolone and Oxymetholone help increase the concentration of the female hormone prolactin. As a result, during the course of these AAS, negative effects reminiscent of estrogenic ones may appear. However, the most serious among progestogenic side effects is a strong inhibition of the HPA axis. This can lead to serious erectile dysfunction and problems with the spermatogenesis process.

Unlike classic gynecomastia, a similar disease caused by a high concentration of prolactin is characterized by more rapid development and serious consequences. Note that during Trenbolone courses, gynecomastia and fluid retention are extremely rare, but athletes often encounter problems with erectile function.

Prolactin inhibitors

Cabergoline

The most effective and popular drug of this class on the modern pharmaceutical market. It is able to selectively act on dopamine type D2 receptors. As a result, prolactin levels decrease in a short time. We recommend taking this drug every fourth day, 0.25 mg. In such a situation, side effects are extremely unlikely.

Bromocreptine

In terms of effectiveness, this drug is not inferior to Cabergoline. However, it has a lot of its own side effects. Among them, we can note a slowdown in the production of endogenous somatotropin. Sometimes with an overdose, an increase in blood pressure is observed. You must remember that prolactin must be present in small quantities in the male body. Thus, it is necessary to use Bromocreptine and Cabergoline in recommended doses.

We recommend that you take tests during the anabolic course to know exactly your hormonal levels. Unfortunately, not every bodybuilding enthusiast is ready for this, including from a financial point of view. In this case, you can follow a few simple rules, the observance of which will minimize the risks of side effects during anabolic cycles:

• The selection of dosages of testosterone-containing AAS must be approached with full responsibility.
• Try not to use Nandrolone, methane and Oxymetholone.
• It is necessary to get acquainted with Trenbolones carefully and carry out the first courses at minimal doses.
• Monitor the condition of the liver and do not start the course until the organ begins to function normally.
• Be sure to do PCT.

Reviews

Athletes who take this substance almost immediately see positive physical and mental effects. There is an increase in muscle mass, fat burning, improvement in mood, general condition, and endurance. Due to excessive dosages, negative factors are observed.

There is a decrease in the level of immunity, lethargy, disturbance of water-salt balance, the appearance of rashes, nausea, sleep disturbance. You need to strictly monitor the dosage and adhere to the norm. Also, these side effects may occur due to sensitivity, an allergic reaction to the components of the drug. Consulting a specialist will help you avoid negative consequences.

Symptoms of increased prolactin during a course of steroids?

Speaking about the growth of prolactin, it is worth mentioning a number of reactions of the body in the case of an increased concentration of this hormone.

Consequences and symptoms of increased prolactin:

• drop in libido;
• headaches, even dizziness;
• fluid retention;
• sleep disturbance;
• apathy;
• gynecomastia;
• obesity;
• galactorrhea (lactation) – the appearance of milk-like fluid from the breast in men;
• severe weakness;
• depression;
• increased appetite;
• acne.